Glimepiride

Glimepiride is oral hypoglycemic agent. It belongs to sulfonylurea class. Glimepiride is chemically identidied as 1-p-2-(3-ethyl-4-methyl-2-oxo-3 pyrroline-1-carboxamido) ethyl-phenylsulfonyl-3-(trans-4-methylcyclohexyl) urea. It was approved by the Food and Drug Administration in 1995 as an adjunct to diet and exercise to lower the blood glucose in patients with type 2 diabetes whose hyperglycemia cannot be controlled by diet and exercise alone.


Brands
PIOTONE GEM PIOTONE GEM GEMPRIDE GEMPRIDE GEMPRIDE GEMPRIDE AMARYL AMARYL AMARYL AMARYL GLIMER GLIMER GLIMER GLIMER GLUCONORMET GLUCONORMET POZE-G POZE-G AGPRIDE AGPRIDE AGPRIDE AGPRIDE GLUCONORM GLUCONORM GLUCONORM GLUCONORM GLOW GLOW GLOW GLOW BROGLIPE BROGLIPE BROGLIPE BROGLIPE LIMORIDE LIMORIDE LIMORIDE LIMORIDE STEADY STEADY STEADY STEADY TAGOZER-G TAGOZER-G TAGOZER-G PIORYL G PIORYL G DIABOLD DIABOLD DIABOLD DIABOLD ORINASE ORINASE ORINASE ORINASE ORINASE MET 2 ORINASE MET 1 GLYPER GLYPER GLYPER GLYPER CAMPRIDE CAMPRIDE CAMPRIDE CAMPRIDE EXEMET EXEMET GLIGUARD GLIGUARD GLOMET GEOPRIDE ZOLIGET ZOLIGET ZOLIGET ZOLIGET ZOLIGET GETFORMIN GETFORMIN GETRYL GETZGLIM GETRYL GETZGLIM GETRYL GETZGLIM GETRYL GETZGLIM EPERIDE NYLORIDE NYLORIDE NYLORIDE NYLORIDE PIOZER G PIOZER G PIOZER G PIOZER G PIOZER G ZEENARYL ZEENARYL ZEENARYL ZEENARYL G-HELIX G-HELIX G-HELIX G-HELIX GENLIP GENLIP GENLIP GENLIP PIOBETIC-G PIOBETIC-G PIOBETIC-G MIPRIDE MIPRIDE GLIBETIC GLIBETIC GLIBETIC PAMARYL PAMARYL PAMARYL PAMARYL GLIO GLIO GLIO GLIO GLIO-P DIATROL DIATROL DIATROL DIATROL MEDIPRIDE MEDIPRIDE MEDIPRIDE MEDIPRIDE GLIP GLIP GLIP NORLIM NORLIM NORLIM NORLIM GLORY GLORY GLORY GLORY BAMARYL BAMARYL GLIOPTIM GLIOPTIM GLIOPTIM GLIOPTIM PIOPRIDE PIOPRIDE EVOPRIDE PLUS EVOPRIDE EVOPRIDE EVOPRIDE EVOPRIDE GLIRIDE GLIRIDE GLIRIDE GLIRIDE PHARPRIDE PHARPRIDE DIALEX AMARIT AMARIT AMARIT AMARIT SUGRAL SUGRAL SUGRAL SUGRAL GPRIDE GPRIDE GPRIDE GPRIDE METME PLUS METME PRABA PRABA PRABA FANTASMIC FANTASMIC FANTASMIC PLUS FANTASMIC PLUS GLYSET GLYSET GLYSET GLYSET G.P.D. G.P.D. G.P.D. G.P.D. GLIMECIDE GLIMECIDE GLIMECIDE GLIMECIDE GAMARYL GAMARYL GAMARYL GAMARYL SUGLOW 3H SUGLOW 3H SUGLOW 3H SUGLOW 3H DIAGLIDE DIAGLIDE SAFGO SAFGO SAFGO SAFGO GLIGO GLIGO GLIGO GLIGO GLIGO-P GLEMEX GLEMEX GLEMEX GLEMEX GLUCORIDE GLUCORIDE CAYPRIDE CAYPRIDE CAYPRIDE CAYPRIDE GLUCOGLIN SUNPRIDE SUNPRIDE DIAGLIM DIAGLIM DIAGLIM DIAGLIM GLIMESCOT GLIMESCOT GLIMESCOT GLIMESCOT GLIMTIDE GLIMTIDE GLIMTIDE NEOGLIM NEOGLIM NEOGLIM NEOGLIM NOARYL NOARYL NOARYL NOARYL MELITUS MELITUS MELITUS MELITUS MEGAPRIDE MEGAPRIDE MEGAPRIDE MEGAPRIDE INITIAL INITIAL INITIAL INITIAL LEADRYL LEADRYL LEADRYL LEADRYL LEA L LEA L LEA L LEA L MELNORM MELNORM MELNORM DAZEMEP DAZEMEP V-PRIDE V-PRIDE V-PRIDE V-PRIDE GLACTIL GLACTIL GLACTIL GLACTIL GLITAMAP PLUS GLITAMAP FORTE GLITAMAP FORTE GLITAMAP GLIBETIC FORTE V PRIDE V PRIDE V PRIDE V PRIDE AGYL AGYL DIFREE OMARID OMARID OMARID OMARID GLIMRYL GLIMRYL GLIMRYL GLIMRYL MEDIRYL MEDIRYL DIBNIL DIBNIL DIBNIL DIBNIL WIPRIDE WIPRIDE GLUNEX GLUNEX GLUNEX GLUNEX G-TAZ GLEMSER GLEMSER GLEMSER A-GLIM A-GLIM RAYPRIDE M RAYPRIDE M RAYPRIDE RAYPRIDE RAYPRIDE RAYPRIDE P RAYPRIDE P RAYPRIDE P RETRYL RETRYL RETRYL RETRYL G-PLUS G-PLUS GLANYL GLANYL GLANYL GLANYL GLIMULIN GLIMULIN GLIMULIN
Adult Dose
Dose: 1 to 2 mg
Single Dose: 1.5 (1.5)
Frequency: 24 hourly
Route: PO
Instructions: Initial
Neonatal
Dose:
Single Dose:
Frequency:
Route:
Instructions: Not recommended in this age group
Paedriatic
Dose:
Single Dose:
Frequency:
Route:
Instructions: Not recommended in this age group
Characteristics
. It is of Synthetic origin and belongs to Sulphonyl Urea. It belongs to Potassium Channel (ATP sensitive) antagonist pharmacological group on the basis of mechanism of action and also classified in Antidiabetic Agent, Sulfonylurea pharmacological group.The Molecular Weight of Glimepiride is 490.60.
Contraindications
Glimepiride is contraindicated in conditions like Diabetic ketoacidosis.
Effects
The severe or irreversible adverse effects of Glimepiride, which give rise to further complications include Thrombocytopenia, Jaundice, Jaundice, Hepatitus, Haumolytic anaemia.The symptomatic adverse reactions produced by Glimepiride are more or less tolerable and if they become severe, they can be treated symptomatically, these include Headache, Anorexia, Diarrhea, Rashes, Urticaria, Epigastric discomfort, Photosensitivity, Nausea and vomiting, Edema, Hypoglycemia, Hyponatremia.
Indications
Glimepiride is primarily indicated in conditions like NIDDM.
Interactions
Glimepiride is known to interact with other drugs, the details of drug interactions is as follows:DrugDetailsSeverityOnsetManagementAescinOxandroloneThe hypoglycemic effect of insulin secretagogues (e.g., sulfonylureas, meglitinides) may be potentiated by certain drugs, including ACE inhibitors, anabolic steroids, fibrates, monoamine oxidase inhibitors (MAOIs), nonsteroidal anti-inflammatory drugs (NSAIDs), salicylates, selective serotonin reuptake inhibitors (SSRIs), sulfonamides, disopyramide, propoxyphene, quinine, and quinidine. These drugs may increase the risk of hypoglycemia by enhancing insulin sensitivity (ACE inhibitors, fibrates); stimulating insulin secretion (salicylates, NSAIDs, disopyramide, quinine, quinidine, MAOIs); increasing peripheral glucose utilization (SSRIs, insulin-like growth factor); and/or inhibiting gluconeogenesis (SSRIs, MAOIs, insulin-like growth factor). Or, they may increase plasma concentration of insulin secretagogues by displacing them from plasma protein binding sites and/or inhibiting their metabolism (fibrates, NSAIDs, salicylates, sulfonamides). Clinical hypoglycemia has been reported during use of these agents alone or with insulin and/or sulfonylureas. Use of SSRIs has also been associated with loss of awareness of hypoglycemia in isolated cases.ModerateClose monitoring for the development of hypoglycemia is recommended if these drugs are coadministered with insulin secretagogues, particularly in patients with advanced age and/or renal impairment. The oral antidiabetic dosage(s) may require adjustment if an interaction is suspected. Patients should be apprised of the signs and symptoms of hypoglycemia (e.g., headache, dizziness, drowsiness, nausea, hunger, tremor, weakness, sweating, palpitations), how to treat it, and to contact their doctor if it occurs. Patients should be observed for loss of glycemic control when these drugs are withdrawn.OxymetholoneThe hypoglycemic effect of insulin secretagogues (e.g., sulfonylureas, meglitinides) may be potentiated by certain drugs, including ACE inhibitors, anabolic steroids, fibrates, monoamine oxidase inhibitors (MAOIs), nonsteroidal anti-inflammatory drugs (NSAIDs), salicylates, selective serotonin reuptake inhibitors (SSRIs), sulfonamides, disopyramide, propoxyphene, quinine, and quinidine. These drugs may increase the risk of hypoglycemia by enhancing insulin sensitivity (ACE inhibitors, fibrates); stimulating insulin secretion (salicylates, NSAIDs, disopyramide, quinine, quinidine, MAOIs); increasing peripheral glucose utilization (SSRIs, insulin-like growth factor); and/or inhibiting gluconeogenesis (SSRIs, MAOIs, insulin-like growth factor). Or, they may increase plasma concentration of insulin secretagogues by displacing them from plasma protein binding sites and/or inhibiting their metabolism (fibrates, NSAIDs, salicylates, sulfonamides). Clinical hypoglycemia has been reported during use of these agents alone or with insulin and/or sulfonylureas. Use of SSRIs has also been associated with loss of awareness of hypoglycemia in isolated cases.ModerateClose monitoring for the development of hypoglycemia is recommended if these drugs are coadministered with insulin secretagogues, particularly in patients with advanced age and/or renal impairment. The oral antidiabetic dosage(s) may require adjustment if an interaction is suspected. Patients should be apprised of the signs and symptoms of hypoglycemia (e.g., headache, dizziness, drowsiness, nausea, hunger, tremor, weakness, sweating, palpitations), how to treat it, and to contact their doctor if it occurs. Patients should be observed for loss of glycemic control when these drugs are withdrawn.SulphamethizoleGlimepiride may be displaced from protein binding sites or their metabolism may be inhibited by some sulfonamides, resulting in increased or prolonged effects or toxicity.Dosage adjustments may be necessary during and after sulfonamide therapy These interactions are sometimes beneficial and sometimes may pose threats to life. Always consult your physician for the change of dose regimen or an alternative drug of choice that may strictly be required.
Interfrence
Risks
Drug should not be given to Pregnant Mothers.If prescribing authority justifies the benefits of the drug against the possible damages he/she should reevaluate them and consult the reference material and previous studies.
Storage
Tab Store Below 40°C. Protect from Sunlight and Heat.
Warnings
Glimepiride should be used with caution in patients with diabetes, kidney disease, liver disease, heart disease or if have any allergy. During times of stress such as fever, infection, injury or surgery, it may be more difficult to control blood sugar, consult the doctor or pharmacist if additional medication may be required. This medication should be used only when clearly needed during pregnancy. Must be taken shortly before meals.
Back to List

Any information that appears on this website page is provided for the purpose of general information. This website has been compiled in good faith by HMIS.Online. However, no guarantee is made as to the completeness, validity or accuracy of the information it contains.